Purpose

A Phase 1, open-label, dose-escalation clinical trial of MBQ-167 in participants with advanced Breast Cancer for whom Standard of Care (SOC) has failed or has proven intolerable.

Conditions

Eligibility

Eligible Ages
Over 21 Years
Eligible Sex
All
Accepts Healthy Volunteers
No

Inclusion Criteria

  • The investigator will evaluate these and other criteria to determine whether a participant can be included in this study. - Histologically and/or cytologically confirmed advanced breast cancer which has progressed after treatment with approved therapies or for which there are no standard therapies available. - Participants with known brain metastases may be eligible if specific conditions are met. - Life expectancy ≥6 months, in the opinion of the investigator, after starting MBQ-167. - Are able to swallow capsules twice daily with a meal.

Exclusion Criteria

  • The investigator will evaluate these and other criteria to determine whether a participant should be excluded from this study. - Inability to take oral medication, or malabsorption syndrome or any other uncontrolled gastrointestinal condition (e.g., nausea, diarrhea, or vomiting) that might impair the bioavailability of MBQ-167. - Females who are pregnant or breastfeeding. - Participants who have received any anticancer treatment within 4 weeks or any investigational agent within 28 days prior to the first dose of trial drug or who have not recovered from any acute toxicity greater than Grade 0 or 1 related to previous anticancer treatment. - Participants who have received any anticancer treatment within 4 weeks or any investigational agent within 28 days prior to the first dose of trial drug or who have not recovered from any acute toxicity greater than Grade 0 or 1 related to previous anticancer treatment. - Active malignancies other than advanced breast cancer will be excluded from the study.

Study Design

Phase
Phase 1
Study Type
Interventional
Allocation
N/A
Intervention Model
Sequential Assignment
Intervention Model Description
Open-label dose escalation following a standard 3+3 cohort design with a 21 day Dose Limiting Toxicity (DLT) evaluation
Primary Purpose
Treatment
Masking
None (Open Label)

Arm Groups

ArmDescriptionAssigned Intervention
Experimental
MBQ-167 oral capsule
A dose ranging from 10mg to 400mg BID following a standard 3+3 cohort design
  • Drug: MBQ-167
    MBQ-167, an inhibitor of Rho GTPases Rac and Cdc42
    Other names:
    • Rac and Cdc42 inhibitor
    • Rac inhibitor
    • Cdc42 inhibitor
    • PAK inhibitor
    • Rac/Cdc42 inhibitor

Recruiting Locations

Precision Next Gen Oncology & Research Center
Beverly Hills, California 90212
Contact:
Rebecca Godin
424-777-0708
RebeccaG@NextGenOnc.com

Florida Cancer Specialists / Sarah Cannon Research Institute / SCRI
Sarasota, Florida 34232
Contact:
Judy S Wang, MD
941-377-9993
jswang@flcancer.com

Sarah Cannon Research Institute/SCRI
Nashville, Tennessee 37203
Contact:
Melissa Sindler
844-482-4812
scri.ddureferrals@scri.com

FDI Clinical Research
San Juan, Puerto Rico 00927
Contact:
Mirelis Acosta-Rivera, MD
(787) 722-1248
info@fdipr.com

More Details

Status
Recruiting
Sponsor
MBQ Pharma

Study Contact

Scott Houston
(415) 404 8838
scott.houston@mbqpharma.com

Detailed Description

The main questions this clinical trial aims to answer are: - What, if any, are the side effects of different dose levels in humans? - What is the maximum tolerated dose? - How does the human body process the drug? - Does the drug slow, stop or eliminate cancer in human participants? Participants will be asked to: - provide informed consent - be evaluated by physicians and provide laboratory specimens to determine if eligible - take MBQ-167 orally twice a day for at least 21 days - may continue dosing, if safe to do so, until not effective or other decision to stop is made - participate in multiple visits that include additional evaluations, laboratory tests and diary review until after stopping the investigational drug

Notice

Study information shown on this site is derived from ClinicalTrials.gov (a public registry operated by the National Institutes of Health). The listing of studies provided is not certain to be all studies for which you might be eligible. Furthermore, study eligibility requirements can be difficult to understand and may change over time, so it is wise to speak with your medical care provider and individual research study teams when making decisions related to participation.