Purpose

The goal of this study is to evaluate nemtabrutinib compared with investigator's choice of ibrutinib or acalabrutinib in participants with chronic lymphocytic leukemia (CLL)/small lymphocytic lymphoma (SLL) who have not received any prior therapy. The primary hypotheses are that (1) nemtabrutinib is non-inferior to ibrutinib or acalabrutinib with respect to objective response rate (ORR) per International Workshop on Chronic Lymphocytic Leukemia (iwCLL) Criteria 2018 by blinded independent central review (BICR) and (2) nemtabrutinib is superior to ibrutinib or acalabrutinib with respect to progression free survival (PFS) per iwCLL Criteria 2018 by BICR.

Conditions

Eligibility

Eligible Ages
Over 18 Years
Eligible Sex
All
Accepts Healthy Volunteers
No

Inclusion Criteria

The main inclusion criteria include but are not limited to the following: - Confirmed diagnosis of CLL/SLL and active disease clearly documented to have a need to initiate therapy. - Has at least 1 marker of disease burden. - Has an Eastern Cooperative Oncology Group (ECOG) performance status of 0 to 2 within 7 days before randomization. - Has the ability to swallow and retain oral medication. - Participants who are hepatitis B surface antigen (HBsAg) positive are eligible if they have received hepatitis B virus (HBV) antiviral therapy for at least 4 weeks and have undetectable HBV deoxyribonucleic acid (DNA) viral load before randomization. - Participants with history of hepatitis C virus (HCV) infection are eligible if HCV ribonucleic acid (RNA) viral load is undetectable at screening. - Participants with human immunodeficiency virus (HIV) who meet ALL eligibility criteria.

Exclusion Criteria

The main exclusion criteria include but are not limited to the following: - Has an active hepatitis B virus/ hepatitis C virus (HBV/HCV) infection. - Has gastrointestinal (GI) dysfunction that may affect drug absorption. - Has diagnosis of Richter Transformation or active central nervous system (CNS) involvement by CLL/SLL. - Has had acquired immune deficiency syndrome (AIDS)-defining opportunistic infection in the past 12 months before screening. - Has clinically significant cardiovascular disease. - Has hypersensitivity to nemtabrutinib or contraindication to ibrutinib or acalabrutinib, or any of the excipients. - Has history of severe bleeding disorder. - Has known additional malignancy that is progressing or has required active treatment within the past 2 years. - Has received any systemic anticancer therapy for CLL/SLL. - Is currently being treated with p-glycoprotein (P-gp) substrates with a narrow therapeutic index, cytochrome P450 3A (CYP3A) strong or moderate inducers or CYP3A strong inhibitors. - Received prior radiotherapy within 2 weeks of start of study intervention, or radiation-related toxicities, requiring corticosteroids. - Received a live or live-attenuated vaccine within 30 days before the first dose of study intervention. Administration of killed vaccines are allowed. - Has received an investigational agent or has used an investigational device within 4 weeks before study intervention administration. - Has active infection requiring systemic therapy, including intravenous (IV) antibiotics during screening. - Participants who have not adequately recovered from major surgery or have ongoing surgical complications.

Study Design

Phase
Phase 3
Study Type
Interventional
Allocation
Randomized
Intervention Model
Parallel Assignment
Primary Purpose
Treatment
Masking
None (Open Label)

Arm Groups

ArmDescriptionAssigned Intervention
Experimental
Nemtabrutinib
Participants will receive nemtabrutinib at specified dose until disease progression, unacceptable toxicity or until discontinuation criteria are met.
  • Drug: Nemtabrutinib
    Administered orally
    Other names:
    • MK-1026
    • ARQ 531
Active Comparator
Ibrutinib/Acalabrutinib
Participants will receive investigator's choice of ibrutinib or acalabrutinib at specified dose until disease progression, unacceptable toxicity or until discontinuation criteria are met.
  • Drug: Ibrutinib
    Administered orally
  • Drug: Acalabrutinib
    Administered orally

Recruiting Locations

USA Mitchell Cancer Institute ( Site 0014)
Mobile 4076598, Alabama 4829764 36604
Contact:
Study Coordinator
888-577-8839

Arizona Oncology Associates - NAHOA ( Site 8007)
Prescott 5309842, Arizona 5551752 86301
Contact:
Study Coordinator
888-577-8839

Alta Bates Summit Medical Center ( Site 0004)
Berkeley 5327684, California 5332921 94704
Contact:
Study Coordinator
888-577-8839

Moores Cancer Center ( Site 0003)
La Jolla 5363943, California 5332921 92093-0698
Contact:
Study Coordinator
888-577-8839

Saint Joseph Hospital ( Site 0026)
Denver 5419384, Colorado 5417618 80218
Contact:
Study Coordinator
303-812-6998

Lutheran Medical Center ( Site 0027)
Golden 5423294, Colorado 5417618 80401
Contact:
Study Coordinator
303-403-3672

Intermountain Health St. Mary's Regional Hospital ( Site 0025)
Grand Junction 5423573, Colorado 5417618 81501
Contact:
Study Coordinator
970-298-7500

Eastern CT Hematology & Oncology Associates ( Site 0033)
Norwich 4839843, Connecticut 4831725 06360
Contact:
Study Coordinator
860-886-8362

Clermont Oncology Center ( Site 0046)
Clermont 4151352, Florida 4155751 34711
Contact:
Study Coordinator
386-538-3169

Florida Cancer Specialists - South ( Site 7001)
Fort Myers 4155995, Florida 4155751 33901
Contact:
Study Coordinator
888-577-8839

Florida Cancer Specialists - East ( Site 7002)
West Palm Beach 4177887, Florida 4155751 33401
Contact:
Study Coordinator
888-577-8839

Parkview Research Center at Parkview Regional Medical Center ( Site 0002)
Fort Wayne 4920423, Indiana 4921868 46845
Contact:
Study Coordinator
260-266-7100

University of Iowa Health Care. ( Site 0017)
Waukee 4880981, Iowa 4862182 50263
Contact:
Study Coordinator
319-356-1616

University of Iowa Health Care. ( Site 0057)
Waukee 4880981, Iowa 4862182 50263
Contact:
Study Coordinator
319-356-1616

Saint Elizabeth Healthcare ( Site 0041)
Edgewood 4290873, Kentucky 6254925 41017
Contact:
Study Coordinator
888-577-8839

Corewell Health-Lemmon Holton Cancer Pavilion ( Site 0011)
Grand Rapids 4994358, Michigan 5001836 49503
Contact:
Study Coordinator
888-577-8839

Regions Hospital ( Site 0042)
Saint Louis Park 5045021, Minnesota 5037779 55416
Contact:
Study Coordinator
952-993-3252

MidAmerica Cancer Care, LLC ( Site 0043)
Kansas City 4393217, Missouri 4398678 64132
Contact:
Study Coordinator
816-974-5050

Intermountain Health St. Vincent Regional Hospital - Cancer Centers of Montana ( Site 0052)
Billings 5640350, Montana 5667009 59102
Contact:
Study Coordinator
406-238-6685

John Theurer Cancer Center at Hackensack University Medical Center ( Site 0016)
Hackensack 5098706, New Jersey 5101760 07601
Contact:
Study Coordinator
888-577-8839

Roswell Park Cancer Institute ( Site 0023)
Buffalo 5110629, New York 5128638 14263
Contact:
Study Coordinator
888-577-8839

Oncology Specialists of Charlotte ( Site 0054)
Charlotte 4460243, North Carolina 4482348 28207
Contact:
Study Coordinator
704-342-1900

Southeastern Medical Oncology Center ( Site 0049)
Goldsboro 4468261, North Carolina 4482348 27534
Contact:
Study Coordinator
919-587-9088

Consultants in Medical Oncology and Hematology (CMOH) ( Site 8002)
Broomall 4556802, Pennsylvania 6254927 19008
Contact:
Study Coordinator
888-577-8839

Cancer Care Associates Of York ( Site 0005)
York 4562407, Pennsylvania 6254927 17403
Contact:
Study Coordinator
888-577-8839

Tennessee Oncology-Chattanooga ( Site 0045)
Chattanooga 4612862, Tennessee 4662168 37404
Contact:
Study Coordinator
615-986-4350

Tennessee Oncology ( Site 0031)
Nashville 4644585, Tennessee 4662168 37203
Contact:
Study Coordinator
615-986-4350

Texas Oncology - Central/South Texas ( Site 8008)
Austin 4671654, Texas 4736286 78705
Contact:
Study Coordinator
888-577-8839

The Center for Cancer and Blood Disorders ( Site 0032)
Fort Worth 4691930, Texas 4736286 76104
Contact:
Study Coordinator
817-759-7013

Texas Oncology - San Antonio ( Site 8006)
San Antonio 4726206, Texas 4736286 78217
Contact:
Study Coordinator
888-577-8839

Texas Oncology - Northeast Texas ( Site 8012)
Tyler 4738214, Texas 4736286 75702
Contact:
Study Coordinator
888-577-8839

University of Virginia Cancer Center ( Site 0040)
Charlottesville 4752031, Virginia 6254928 22903
Contact:
Study Coordinator
434-243-2649

Inova Schar Cancer Institute ( Site 0015)
Fairfax 4758023, Virginia 6254928 22031
Contact:
Study Coordinator
888-577-8839

Virginia Commonwealth University (VCU) Medical Center ( Site 0030)
Richmond 4781708, Virginia 6254928 23298
Contact:
Study Coordinator
804-628-2072

Medical Oncology Associates, PS (dba Summit Cancer Centers) ( Site 0010)
Spokane 5811696, Washington 5815135 99208
Contact:
Study Coordinator
888-577-8839

SSM Health Dean Medical Group - South Madison Campus Health Research/Circuit Clinical ( Site 0048)
Madison 5261457, Wisconsin 5279468 53715
Contact:
Study Coordinator
608-410-2700

University Hospital and UW Health Clinics ( Site 0006)
Madison 5261457, Wisconsin 5279468 53792
Contact:
Study Coordinator
888-577-8839

More Details

Status
Recruiting
Sponsor
Merck Sharp & Dohme LLC

Study Contact

Toll Free Number
1-888-577-8839
Trialsites@msd.com

Notice

Study information shown on this site is derived from ClinicalTrials.gov (a public registry operated by the National Institutes of Health). The listing of studies provided is not certain to be all studies for which you might be eligible. Furthermore, study eligibility requirements can be difficult to understand and may change over time, so it is wise to speak with your medical care provider and individual research study teams when making decisions related to participation.